Search Result "MDCK-MDR1"


Evaluating Potential P-gp Substrates: Main Aspects to Choose the Adequate Permeability Model for Assessing Gastrointestinal Drug Absorption

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 15 Issue: 10 Year: 2015 Page: 858-871
Author(s): Joao Batista da Silva Junior,Thaisa Marinho Dezani,Andre Bersani Dezani,Cristina Helena dos Reis Serra

An MDR-EGFP Gene Fusion Allows for Direct Cellular Localization, Function and Stability Assessment of P-Glycoprotein

Journal: Current Drug Delivery
Volume: 1 Issue: 1 Year: 2004 Page: 43-56
Author(s): Jordi Petriz, Michael M. Gottesman, Josep M. Aran

Interaction of Probenecid with the Breast Cancer Resistance Protein Transporter (BCRP/ABCG2)

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 4 Year: 2006 Page: 236-241
Author(s): G. Merino, R. Real, A. J. Molina, M. M. Pulido, J. G. Prieto, A. I. Alvarez

Role of P-glycoprotein in the Transport of Tanshinone I, One Active Triterpenoid from Salvia miltiorrhiza

Journal: Drug Metabolism Letters
Volume: 2 Issue: 3 Year: 2008 Page: 223-230
Author(s): Xing-Xiao Li, Zhi-Wei Zhou, Shu-Feng Zhou

Opioid Transport by ATP-Binding Cassette Transporters at the Blood-Brain Barrier: Implications for Neuropsychopharmacology

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 2 Year: 2011 Page: 2829-2842
Author(s): Nicolas Tournier, Xavier Decleves, Bruno Saubamea, Jean-Michel Scherrmann, Salvatore Cisternino

Current Frontiers

The Tetrahydroisoquinoline Scaffold in ABC Transporter Inhibitors that Act as Multidrug Resistance (MDR) Reversers

Journal: Current Topics in Medicinal Chemistry
Volume: 22 Issue: 31 Year: 2022 Page: 2535-2569
Author(s): Maria Novella Romanelli

Role of Microfluidics in Blood-Brain Barrier Permeability Cell Culture Modeling: Relevance to CNS Disorders

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 15 Issue: 3 Year: 2016 Page: 301-309
Author(s): Alexander L. Rusanov,Natalia G. Luzgina,George E. Barreto,Gjumrakch Aliev

Two Branched Polar Groups and Polar Linker Moieties of Thiophene Amide Derivatives Are Essential for MRP2/ABCC2 Recognition

Journal: Drug Metabolism Letters
Volume: 4 Issue: 4 Year: 2010 Page: 254-261
Author(s): Yiding Hu, Kathleen E. Sampson, Li Xing, Na Li, Bruce R. Heyde, Jin Xie, Yurong Lai

Utility of Mdr1-Gene Deficient Mice in Assessing the Impact of P-glycoprotein on Pharmacokinetics and Pharmacodynamics in Drug Discovery and Development

Journal: Current Drug Metabolism
Volume: 4 Issue: 4 Year: 2003 Page: 272-291
Author(s): Cuiping Chen, Xingrong Liu, Bill J. Smith

Inhibition of Hepatobiliary Transporters by A Novel Kinase Inhibitor Contributes to Hepatotoxicity in Beagle Dogs

Journal: Drug Metabolism Letters
Volume: 7 Issue: 1 Year: 2013 Page: 15-22
Author(s): John Scott Daniels,Yurong Lai,Sarah South,Po-Chang Chiang,Daniel Walker,Bo Feng,Rouchelle Mireles,Laurence O. Whiteley,Jeremy W. Mckenzie,Jeffrey Stevens,Robert Mourey,David Anderson,John W. Davis II

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